Contact Us
Order Status
Certificates of Analysis
Safety Data Sheets
Select Country

Please select a country, so we can supply you with the most accurate content available for your country or region.

  • Compare Products
  • Sign In / Register
    • My Quote
    Cart
    Order Status
    main product photo

    Elastatinal, ≥50%, 1 mg

    In stock

    SKU:  0215284701

    Synonyms
    (2S)-2-[(4S)-2-Amino-1,4,5,6-tetrahydro4-pyrimidinyl]-N-[[[(1S)-1-carboxy-3-methylbutyl]amino]carbonyl]glycyl-N1-[(1S)-1-methyl-2-oxoethyl-L-glutamamide; N-(Nα-Carbonyl-Cpd-Gln-Ala-al)-Leu where Cpd = capreomycidine = (S,S)-α-[2-Iminohexahydro-4-pyrimidylglycine]
    CAS Number:
    51798-45-9
    Molecular Formula:
    C21H36N8O7
    Molecular Weight:
    512.57
    Beilstein Registry Number:
    873543
    EC Number:
    257-426-7
    Packaging size:
    1 mg
    Contact Us for Specific Delivery Information
    Request A Custom or Bulk Quote
    Specifications
    SKU 0215284701
    Alternate Names (2S)-2-[(4S)-2-Amino-1,4,5,6-tetrahydro4-pyrimidinyl]-N-[[[(1S)-1-carboxy-3-methylbutyl]amino]carbonyl]glycyl-N1-[(1S)-1-methyl-2-oxoethyl-L-glutamamide; N-(Nα-Carbonyl-Cpd-Gln-Ala-al)-Leu where Cpd = capreomycidine = (S,S)-α-[2-Iminohexahydro-4-pyrimidylglycine]
    Base Catalog Number 15284701
    Beilstein Registry Number 873543
    Biochemical Physiological Actions Potent, irreversible elastase inhibitor (Ki = 240 nM). Elastatinal is a much stronger inhibitor of elastase from pancreas than from leucocytes. Elastatinal is a strong competitive inhibitor of elastase which is found in some species of Streptomyces, showing 50% inhibition at 0.29 ug/mL, while greater than 250 ug/mL is required for other proteases.
    CAS # 51798-45-9
    EC Number 257-426-7
    Extinction Coefficient E1% = 1.5 (0.1 N HCl), 2.5 (0.1 M phosphate, pH 7.0)(Lit.)
    Molecular Formula C21H36N8O7
    Molecular Weight 512.57
    Pack Size 1 mg
    Personal Protective Equipment Eyeshields, Gloves, respirator filter
    pKa 3.7 and >10.5 (Lit.)
    Purity ≥50%
    RTECS Number LZ9600000
    Solubility Soluble in water (20 mg/mL - clear solution), DMSO, or methanol. Also soluble in pyridine, dimethyl sulfoxide, and slightly soluble in ethanol.
    Typical Working Concentration Effective concentration is typically 0.5 to 2 ug/mL.
    Usage Statement Unless specified otherwise, MP Biomedical's products are for research or further manufacturing use only, not for direct human use. For more information, please contact our customer service department.
    UV Visible Absorbance λmax: 275 nm, 298 nm (Lit.)
    Documents

    Certificate of Analysis (COA)

    MP COA [152847] lot ID: QR13515 MP COA [152847] lot ID: QR13515

    Datasheet

    Datasheet
    DS [02152847] DS [02152847]